Mu kutupa ndi tizilombo toyambitsa matenda osadziwika kapena tizilombo toyambitsa matenda (tizilombo toyambitsa matenda), mankhwala osokoneza bongo omwe ali ndi ntchito yaikulu kwambiri. 5-NOC ndi wothandizira odwala antibacterial ogwira ntchito motsutsana ndi tizilombo todziwika kwambiri. Ndizotsutsana ndi mazira ena.
5-NOC - yopangidwa
Chofunika chachikulu cha mankhwalawa mu funso ndi nitroxoline. Ndicho chigawo chochokera ku 8-hydroxyquinoline, chomwe chimalepheretsa kufotokoza kwa DNA kuchokera ku maselo a tizilombo ndipo timalepheretsa kubereka. Zothandizira zothandizira zomwe zikuphatikizidwa mu mapepala a 5-NOC-mapepala ndi awa:
- lactose monohydrate;
- calcium hydrogen phosphate;
- chimanga cha chimanga;
- Povidone K25;
- colloidal silicon dioxide;
- talc woyera;
- magnesium stearate;
- crospovidone.
Mapiritsi amapangidwa mu chipolopolo choteteza, chomwe chili ndi zinthu zotsatirazi:
- carmellose sodium;
- chithandizo;
- colloidal silicon dioxide;
- Povidone K25;
- titaniyamu dioxide;
- chimanga cha chimanga;
- sucrose;
- talc woyera;
- calcium carbonate;
- Mitundu ya zakudya - chikasu "Sunset Sunset" (E110) ndi quinoline (E104).
5-NOC - chizindikiro
Mankhwalawa amapangidwa pofuna kuchiza matenda opatsirana kapena ocheperako omwe amapezeka m'makina ndi kubereka. Mapiritsi 5-NOC ndi othandiza polimbana ndi magulu a tizilombo:
- Gram-positive aerobic ndi anaerobic;
- ger-negative aerobic ndi anaerobic;
- mycoplasma ;
- ureaplasma ;
- Trichomonas;
- Mycobacterium chifuwa chachikulu;
- dermatophytes;
- nkhungu nkhungu;
- wosankhidwa;
- Tizilombo ta tizilombo toyambitsa matenda omwe amachititsa kuti mycoses ayambe kwambiri.
5-NOC - zizindikiro zogwiritsidwa ntchito:
- cystitis;
- pyelonephritis ;
- epididymitis;
- urethritis;
- Matenda a adenoma, carcinoma a prostate;
- prostatitis;
- Kutupa koyambitsa mkodzo kapena kapezi.
Chofotokozedwa chokonzekera chimagwiritsidwa ntchito popewera matenda m'madera otere:
- nthawi yopuma;
- kuchiritsa matenda;
- chithunzithunzi ;
- catheterization.
5-NOC - zotsatira
Mankhwala olimbana ndi antibacterial angapangitse kuti thupi lisamachite chilichonse. Izi zikutanthauza kuti kawirikawiri zimatsogolera ku zotsatira. Milandu yapadera, kukonza 5-NOC kumayambitsa:
- tachycardia;
- kusanza;
- anorexia;
- chisokonezo;
- wosalimba chiwindi ntchito;
- chizungulire;
- optic neuritis (ndi kuvomereza kwa nthawi yaitali);
- paresthesia;
- kusowa mgwirizano;
- mutu;
- mapuloteni;
- chithandizo;
- kuwonjezeka kwa uric acid;
- urticaria;
- kuyabwa kwa khungu;
- ataxia;
- kuwonetsa mkodzo mu utoto wobiriwira.
5-NOC zotsutsana
Chida ichi sichivomerezedwa chifukwa chosagwirizana pakati pa zosakaniza zomwe zili pamwambapa, kuphatikizapo mankhwala othandizira ndi zigawo zina. Mankhwala 5-NOC amatsutsana pazifukwa izi:
- mimba;
- chowongolera;
- kuyamwitsa;
- Kusokonezeka kwakukulu kwa chiwindi kapena impso zokhala ndi mphamvu zopangidwa ndi creatinine zosachepera 20ml / min (zolembedwa kawirikawiri, mosamala);
- ali ndi zaka zitatu.
Kodi mungatenge mapiritsi asanu ndi awiri a NOC?
Gawo la tsiku ndi tsiku la mankhwala limadalira zaka komanso kukhalapo kwa matenda ena aakulu. Akuluakulu pa tsiku amafunika 400 mg ya mankhwala 5-NOC - kugwiritsa ntchito kumaphatikizapo kutenga mlingowu, magawo 4, 100 mg (mapiritsi awiri) musanadye. Ndi tizilombo toyambitsa matenda, gawoli laphatikizidwa (800 mg). Ana oposa zaka zisanu amalamulidwa 200-400 mg ya mankhwala maola 24, ndipo ana a zaka 3-5 - 200 mg. Njira yowonjezereka ya mankhwala siidapitirira milungu 2-4, ngati kuli kotheka, kubwereza.
Ngati mulibe vutoli, 5-NOC imagwiritsidwa ntchito mosamala kwambiri - zizindikiro zosagwiritsidwa ntchito siziphatikizapo matendawa, koma pa matenda aakulu, antibiotic imatha kulamulidwa. Pazochitikazi, tenga 1 piritsi limodzi 4 pa tsiku. Ndikofunika kufufuza nthawi zonse momwe impso ndi chiwindi zimayendera ndikuchiza ndikuyang'ana momwe mulingo umayendera.
5-NOC - ntchito ya cystitis
Mlingo wa wothandizira ma antimicrobial ali ndi mlingo woyenera wa 400 mg nitroxoline maola 24 alionse. 5-NOC ndi cystitis ikulimbikitsidwa njira ya masiku 10-21. Nthawi yeniyeni ya mankhwala imayesedwa ndi wa urologist wochokera ku mayeso a labotale, kuuma kwa njira yotupa, ndi kukhalapo kwa zotsatira za mankhwala. Nthawi zina ziyenera kupitilira kwa mwezi umodzi, makamaka ngati matendawa akuphatikizidwa kapena wachiwiri.
5-NOC ndi pyelonephritis
Omwe akufotokozedwa kuti matendawa ali ndi mawonekedwe ovuta amafunika njira yaying'ono yothandizira maantibayotiki, 400 mg tsiku lililonse kwa milungu 2-2.5. Mu nthawi yambiri ya pyelonephritis, wothandizira uroji amalingalira momwe angatengere 5-NOC. Pali ndondomeko ya chithandizo chamkati chamkati (2-3 miyezi 14) komanso mitundu yambiri yogwiritsira ntchito mankhwalawa mu 100 mg mg.
Nthawi zina zimatengera kulandira kwautali kwambiri kwa 5-NOC - zizindikiro zogwiritsidwa ntchito zikuphatikizapo mitundu yosiyanasiyana ya pyelonephritis:
- zitsulo;
- purulent;
- zowerengeka.
5-NOC mukutenga
Pa nthawi yonse yowonongeka, njira yodzikongoletsera yazimayi imakhala yotetezeka kwambiri ndipo imakhala yotsekemera. Chifukwa cha ichi, amayi omwe akuyembekezera nthawi zambiri amakhala ndi chidwi ndi 5-NOC - ndingathe kumwa madziwa panthawi yomwe ali ndi mimba komanso mlingo uliwonse. Mankhwalawa amatsutsana ndi izi, chifukwa zingasokoneze chitukuko kapena kupanga mwanayo.
5-NOC ofanana
Pamene mankhwalawa akugwiritsa ntchito mankhwala osokoneza bongo sangagwiritsidwe ntchito kapena amachititsa mavuto aakulu, ayenera kuchotsedwa. Njira yokhayo yothetsera mapiritsi asanu ndi awiri-NOC ndi kugwiritsa ntchito zizindikiro zofanana kapena zowonjezera. Pali zifaniziro ziwiri zodziwika kwa mankhwala omwe akufotokozedwa:
- Nitroxoline (Germany, Russia);
- Uroksolin (Ukraine).
Mankhwala oyamba amapangidwa ndi mankhwala osiyanasiyana, omwe ali othandizira kuchipatala. Njira yachiwiri yothetsera imakhala mu mapiritsi omwe ali ndi mankhwala okhudzana ndi 50 mg. Ngati kusagwirizana kwa nitroxoline kapena zochokera kumtundu wake, ndikofunika kugwiritsa ntchito generic. Mankhwalawa ali ndi makhalidwe ofanana ndi 5-NOC - zizindikiro zazikulu zogwiritsiridwa ntchito, antibacterial ndi antitifungal ntchito, koma zosiyana. Mankhwala othandiza amawoneka ngati bacteriophages:
- kamwazi kakang'ono;
- zosangalatsa;
- ngati;
- staphylococcal;
- Mapuloteni;
- Klebsiella chibayo;
- Pseudomonas (pseudomonas);
- kolik-proteyny;
- salmonella.
Zowonjezera zina ndi zizindikiro zofanana:
- Fosmicin;
- Ureacid;
- Zosokoneza;
- Bernie;
- Fosmicin;
- Chithunzi;
- Phosphoral;
- Urophosfabol;
- Chisokonezo;
- Kupanga;
- Urofoscin;
- Phosphocin;
- Espa-Focine.